1. Product Overview & Specifications

2-Amino-5-Fluoro-4-Picoline (CAS 1002341-50-4) is a fluorinated pyridine derivative with molecular formula C₆H₆FN₂. Key parameters:

Comparative Analysis

2. Key Applications

Pharmaceutical Intermediates

Used in synthesis of kinase inhibitors and anticancer agents due to fluorine’s electronegativity enhancing binding affinity.

Agrochemicals

Critical for creating fluorinated pesticides with improved metabolic stability and bioavailability.

3. Usage Scenarios

Scenario 1: Anticancer Drug Development

Used as a building block in EGFR inhibitor synthesis at 0.5-2 mol% loading, achieving 85% yield in Suzuki-Miyaura couplings.

4. Client Case Studies

Case 1: PharmaGen Solutions

Challenge: Required high-purity fluorinated intermediate for PI3K inhibitor R&D.
Solution: Used 2-Amino-5-Fluoro-4-Picoline (98.7% purity) in Buchwald-Hartwig reactions.
Result: Reduced synthesis steps from 5 to 3, saving 22% in production costs.

Case 2: AgroChem Innovations

Developed next-gen fungicide using our compound as key intermediate, achieving 40% longer field persistence vs non-fluorinated analogs.

5. Inquiry & Contact

Request pricing, COA, or custom synthesis options:
Email: info@vivalr.com
Tel: (86) 15866781826

Why Choose Us:
– Batch-to-batch consistency (RSD <0.8%)
– Custom fluorination services available
– ISO 9001-certified production