nafamostat mesilate cas 82956-11-4

Chemical Name:Nafamostat mesilate
CAS No.:82956-11-4
Molecular weight:539.58
Appearance:White crystalline powder
Assay: 98% min

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Nafamostat Mesilate (CAS 82956-11-4) Ultimate User Guide

Table of Contents

1. Product Specifications & Comparative Analysis

Parameter Specification Vivalr Standard Competitor A
CAS Number 82956-11-4 Identical
Purity ≥99.2% HPLC Verified ≥98.5%
Molecular Formula C19H17N3O4S Consistent
Storage 2-8°C Desiccated Stability Guaranteed Ambient Allowed

2. Clinical & Industrial Applications

Primary Therapeutic Uses:

  • Protease Inhibition: Serine protease inhibitor targeting thrombin/trypsin
  • Anticoagulant Therapy: Extracorporeal circulation anticoagulation
  • COVID-19 Treatment: TMPRSS2 protease inhibition
  • Pancreatitis Management: Trypsin activity suppression

3. Professional Usage Guidelines

Application Concentration Range Solvent Compatibility
In Vitro Coagulation Studies 0.1-1 μM PBS/Saline
Viral Entry Inhibition 5-10 μM Cell Culture Medium
Animal Studies 0.3 mg/kg Sterile Water

4. Verified Application Cases

Case 1: COVID-19 Research (University of Tokyo)

Application: Viral entry inhibition in human lung cells
Result: 78% reduction in viral load at 7μM concentration
Technical Support: Custom purity optimization

Case 2: Acute Pancreatitis Treatment (ABC Pharma)

Application: Drug formulation development
Outcome: Phase II clinical trial approval
Batch Consistency: 99.1-99.4% purity across 15 batches

Case 3: Hemodialysis Anticoagulation (Berlin Medical Center)

Usage: Alternative to heparin in 120 patients
Results: 92% efficacy with reduced bleeding risk
Dosage: 0.25 mg/kg/hr during procedures

5. Technical Consultation & Ordering

Contact Our Experts:

Email: info@vivalr.com
Phone: (86) 15866781826

Request Information:

  • Custom synthesis options
  • GMP-grade manufacturing
  • Bulk pricing (1kg+ orders)
  • Regulatory documentation

FAQ Section

Q: Solubility in DMSO?
A: 50 mg/mL with gentle warming

Q: Stability in solution?
A: 24hr stability at 4°C

Q: International shipping?
A: DHL/FedEx with cold chain

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