Atipamezole HCL CAS 104075-48-1

Chemical Name: Atipamezole HCL
CAS No.: 104075-48-1
Molecular Formula: C14H16N2.HCl
Molecular weight: 248.75
Appearance: White powder
Assay: 98%min

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Atipamezole HCl CAS 104075-48-1: Comprehensive Guide for Veterinary Applications

Table of Contents

1. Product Overview & Specifications

Chemical Name: Atipamezole Hydrochloride
CAS Number: 104075-48-1
Molecular Formula: C14H16N2O·HCl
Purity: ≥99% (HPLC)
Appearance: White crystalline powder

Comparative Analysis

Parameter Atipamezole HCl Yohimbine HCl Flumazenil
Reversal Target α2-Adrenoceptor Agonists α2-Adrenoceptors Benzodiazepines
Onset Time 5-15 minutes 15-30 minutes 1-2 minutes
Duration 2-4 hours 3-6 hours 45-90 minutes

2. Key Applications & Use Cases

Primary Veterinary Uses

  • Reversal of medetomidine/dexmedetomidine sedation
  • Emergency treatment for α2-agonist overdose
  • Post-operative recovery acceleration

Emerging Applications

  • Zoological park animal management
  • Wildlife conservation sedation protocols
  • Research animal anesthesia recovery

3. Usage Guidelines & Best Practices

Dosing Protocol

Species Dose (μg/kg) Administration Route
Canine 50-100 IM/IV
Feline 75-150 IM
Equine 30-60 IV

Critical Considerations

  • Monitor cardiovascular parameters during reversal
  • Contraindicated in animals with heart disease
  • Store at 2-8°C protected from light

4. Industry Case Studies

Emergency Clinic Implementation

Challenge: Prolonged recovery in critical care patients
Solution: Atipamezole HCl protocol implementation
Outcome: 40% reduction in ICU occupancy time

Wildlife Research Application

Project: Brown bear conservation in Scandinavia
Usage: Field anesthesia reversal agent
Result: 95% safe recovery rate in 156 procedures

5. Client Implementation Examples

Veterinary Hospital Chain (North America)

  • 18 locations standardized reversal protocols
  • Reduced post-op complications by 28%
  • Improved surgical throughput capacity

Pharmaceutical Manufacturer (EU)

  • Integrated into pre-clinical trial protocols
  • Enhanced animal welfare compliance
  • Accelerated drug development cycles

6. Request Customized Solutions

Contact our veterinary pharmacology experts:
Email: info@vivalr.com
Phone: (86) 15866781826

Request:

  • Custom dosage formulations
  • Species-specific protocol development
  • Bulk purchasing agreements
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