4-(4-Aminobenzyl)piperazine-1-carboxylic acid tert-butyl ester: Comprehensive User Guide
Table of Contents
1. Product Overview & Comparative Analysis
Key Specifications
Parameter | Specification |
---|---|
CAS Number | 147083-93-0 |
Molecular Formula | C17H25N3O2 |
Molecular Weight | 303.41 g/mol |
Purity | ≥98% (HPLC) |
Appearance | White to off-white crystalline powder |
Competitive Benchmarking
Feature | Our Product | Generic Alternatives |
---|---|---|
Boc Protection Stability | Stable up to 12 months at 2-8°C | 6-8 months typical |
Aminobenzyl Reactivity | Controlled orientation for selective coupling | Randomized coupling common |
Pharma-Grade Certification | ISO 9001:2015 compliant | Limited documentation |
2. Detailed Applications
Pharmaceutical Intermediates
Enables precise synthesis of:
- Kinase inhibitor scaffolds
- GPCR-targeted compounds
- Anticancer drug candidates
Chemical Biology Probes
- Amine-reactive conjugation sites
- Controlled release via Boc deprotection
3. Usage Scenarios & Case Studies
Case Study A: Antiviral Drug Development
Challenge: Achieve >95% coupling efficiency in nucleoside analog synthesis
Solution: Utilized aminobenzyl group for directed ortho-metalation
Outcome: 97.3% yield with 99.1% purity
Case Study B: PET Tracer Synthesis
Challenge: Radiolabeling efficiency below 80%
Solution: Boc protection prevented amine interference
Outcome: 89% radiochemical yield achieved
4. Client Success Stories
Global Pharma Leader (Top 10 Innovator)
Application: JAK2 inhibitor scale-up
Results: Reduced synthesis steps from 7 to 4
Testimonial: "Critical for our Phase III candidate manufacturing"
Biotech Startup (CNS Focus)
Application: Dopamine D3 receptor modulator
Results: 40% cost reduction in lead optimization
Testimonial: "Accelerated our IND submission timeline"
5. Request Customized Solutions
Contact our technical team for:
- Bulk pricing (1kg+ quantities)
- Custom purity profiles (up to 99.9%)
- Regulatory support (DMF filings)
Email: info@vivalr.com
Phone: (86) 15866781826