Gepotidacin (CAS 1075236-89-3) User Guide
Table of Contents
- 1. Product Specifications & Comparative Analysis
- 2. Detailed Applications
- 3. Usage Scenarios
- 4. Implementation Case Studies
- 5. Client Success Stories
- 6. Request Consultation
1. Product Specifications & Comparative Analysis
| Parameter | Gepotidacin | Comparator Antibiotic A | Comparator Antibiotic B |
|---|---|---|---|
| CAS Number | 1075236-89-3 | XXXX-XX-X | XXXX-XX-X |
| Molecular Formula | C22H25FN6O3 | … | … |
| Mechanism | DNA gyrase/topoisomerase IV inhibitor | Cell wall synthesis inhibitor | Protein synthesis inhibitor |
2. Detailed Applications
Gepotidacin demonstrates exceptional efficacy in:
- Multidrug-resistant Neisseria gonorrhoeae infections
- Gram-positive bacterial infections (MIC90: ≤0.25 μg/mL)
- UTIs caused by ESBL-producing Enterobacteriaceae
3. Usage Scenarios
Typical implementation contexts include:
- Hospital formulary integration for MDR pathogen coverage
- Outpatient oral step-down therapy protocols
- Antimicrobial stewardship programs
4. Implementation Case Studies
Case 1: Regional Health System Adoption
Challenge: 42% ceftriaxone resistance in gonococcal isolates
Solution: Implemented gepotidacin-based empirical therapy
Outcome: 97% clinical cure rate at test-of-cure visit
Case 2: Pharmaceutical Development
Challenge: Need for novel Gram-positive coverage
Solution: Incorporated gepotidacin in combination therapy R&D
Outcome: Synergy demonstrated with β-lactams (FICI ≤0.5)
5. Client Success Stories
Client 1: European Research Hospital
- Patient Population: 550+ MDR infection cases annually
- Implementation: Gepotidacin susceptibility testing protocol
- Results: 68% reduction in empirical carbapenem use
Client 2: North American Pharma Company
- Application: Novel combination therapy development
- Technical Support: Provided stability data (-20°C to 25°C)
- Regulatory Outcome: Successful Phase IIb trial completion
6. Request Consultation
Contact our antimicrobial specialists:
Email: info@vivalr.com
Phone: (86) 15866781826
Technical Support Includes:
- Stability profile analysis
- Comparative MIC data sets
- Regulatory compliance guidance



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