4-Amino-5-ethylsulfonyl-2-methoxybenzoic Acid: Comprehensive User Guide
Table of Contents
1. Product Overview & Specifications
| Parameter | Details |
|---|---|
| Chemical Formula | C10H13NO5S |
| Molecular Weight | 259.28 g/mol |
| CAS Number | 4840-63-5 |
| Appearance | White to off-white crystalline powder |
| Purity | ≥98% (HPLC) |
2. Key Applications
This compound serves as a critical intermediate in the synthesis of Amisulpride, a potent antipsychotic agent. Its unique structural features enable:
- Selective dopamine D2/D3 receptor antagonism
- Enhanced bioavailability in API formulations
- Controlled release properties in sustained-action medications
3. Usage Scenarios
Pharmaceutical Synthesis Workflow
- Methylation: Reacts with dimethyl sulfate under controlled pH
- Sulfonation: Bromine/thiocyanate-mediated functionalization
- Ethylation: KOH-catalyzed alkylation with bromoethane
- Oxidation: H2O2-driven sulfone formation
4. Client Case Studies
Case Study 1: European Pharma Innovator
Challenge: Scaling Amisulpride production while maintaining ≤0.1% impurity levels
Solution: Implemented our GMP-grade batch with 24.5% total synthesis yield
Outcome: Achieved 99.2% API purity, reducing purification costs by 18%
Case Study 2: Asian Research Consortium
Challenge: Developing novel dopamine modulators
Solution: Custom functionalization of the methoxy-sulfone moiety
Outcome: 3 patent filings for CNS-targeted therapeutics
5. Technical Support & Inquiries
For batch specifications, MSDS, or custom synthesis requirements:
| Email: | info@vivalr.com |
| Phone: | (86) 15866781826 |


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