Semaglutide (CAS 910463-68-2): Comprehensive Product Guide
Table of Contents
1. Product Specifications & Comparative Analysis
| Parameter | Semaglutide | Alternative GLP-1 Agonists |
|---|---|---|
| CAS Number | 910463-68-2 | N/A |
| Molecular Formula | C187H291N45O59 | Varies by compound |
| Molecular Weight | 4113.58 g/mol | 2,500-4,500 g/mol |
| Administration Forms | Subcutaneous injection (Ozempic/Wegovy) Oral tablet (Rybelsus) |
Primarily injectable |
| Half-Life | 165 hours | 11-13 hours (short-acting analogs) |
2. Clinical Applications
Primary Indications
- Glycemic control in Type 2 Diabetes Mellitus (HbA1c reduction up to 1.8%)
- Chronic weight management (BMI ≥30 kg/m² or ≥27 kg/m² with comorbidities)
- Cardiovascular risk reduction in diabetic patients
Emerging Applications
- Non-alcoholic steatohepatitis (NASH) management
- Chronic kidney disease progression delay
- Neurodegenerative disorders research (Alzheimer’s/Dementia)
- Addiction medicine (alcohol dependence trials)
3. Usage Guidelines
Dosing Protocol
| Formulation | Initial Dose | Maintenance Dose | Administration |
|---|---|---|---|
| Ozempic® (injection) | 0.25 mg weekly | 0.5-2.0 mg weekly | Subcutaneous (abdomen/thigh) |
| Rybelsus® (oral) | 3 mg daily | 7-14 mg daily | Fasting state (30 min pre-meal) |
| Wegovy® (obesity) | 0.25 mg weekly | 2.4 mg weekly | Subcutaneous |
4. Adverse Effects & Safety
Common Reactions (≥10%)
- Nausea (44%)
- Diarrhea (30%)
- Vomiting (24%)
Black Box Warnings
- Thyroid C-cell tumor risk (rodent studies)
- Contraindicated in Multiple Endocrine Neoplasia syndrome type 2
FDA Updates (2023)
- Added ileus/intestinal obstruction risk (0.8% incidence)
- Pancreatitis monitoring requirements
5. Client Success Stories
Case 1: Pharmaceutical Manufacturer
Client: Novo Nordisk A/S
Application: Diabetes management formulation
Outcome: Achieved $29.3B annual revenue (2024) with Ozempic®
Case 2: Research Institution
Client: University of North Carolina
Application: Addiction medicine trials
Outcome: Phase II trials showing 40% alcohol craving reduction
Case 3: Healthcare Provider
Client: Mayo Clinic Endocrinology Division
Application: Obesity management program
Outcome: 15.3% mean body weight loss over 68 weeks
6. Request Consultation
For clinical protocols, bulk procurement, or research collaboration:
Email: info@vivalr.com
Tel: (86) 15866781826



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