5-FORMYL-2,4-DIMETHOXYPYRIMIDINE

5-FORMYL-2,4-DIMETHOXYPYRIMIDINE: Technical Guide & Application Insights

Table of Contents

• Product Overview
• Specifications & Comparative Analysis
• Key Applications
• Usage Guidelines
• Industry Case Studies
• Contact for Technical Consultation

Product Overview

5-FORMYL-2,4-DIMETHOXYPYRIMIDINE (CAS 943319-16-8) is a high-purity heterocyclic compound with molecular formula C₇H₈N₂O₃ and molecular weight 168.15 g/mol. This yellow crystalline powder exhibits:

• Melting Point: 156-158°C
• Solubility: DCM > DMF > THF
• Storage: -20°C protected from light

Specifications & Comparative Analysis

Key Applications

1. Pharmaceutical Intermediate

Critical building block for:

• EGFR tyrosine kinase inhibitors
• Anticancer prodrugs (≥85% yield improvement vs traditional routes)
• Antiviral nucleotide analogs

2. Agrochemical Development

Enables synthesis of:

• Systemic fungicides with EC₅₀ ≤ 0.5 ppm
• Neonicotinoid alternatives

Usage Guidelines

Industry Case Studies

Case 1: Oncology Drug Development

Client: Top 10 Global Pharma Company
Challenge: Improve third-generation TKI synthesis efficiency
Solution: Used as key intermediate in Pd-catalyzed cross-couplings
Result: 40% reduction in step count, 92% overall yield

Case 2: Green Pesticide Innovation

Client: EU Agrochemical Innovator
Application: Novel insect growth regulator
Performance: LC₅₀ 2.3 μg/mL against target pests

Technical Consultation & Sampling

For formulation support, custom synthesis, or bulk pricing:

Email: info@vivalr.com
Tel: (86) 15866781826

Request SDS, COA, or application notes:

• GMP-grade batches available
• Custom functionalization services