Chemical Name: Fexinidazole
Synonyms: 1-Methyl-2-[[4-(methylthio)phenoxy]methyl]-5-nitro-1H-imidazole; HOE-239
CAS No.: 59729-37-2
Molecular Formula: C12H13N3O3S
Molecular Weight: 279.31
Appearance: Crystal
Parameter | Specification |
---|---|
IUPAC Name | 1-Methyl-2-nitro-5-(1-methyl-5-nitro-1H-imidazol-2-yl)-1H-imidazole |
Molecular Formula | C10H11N5O4 |
Molecular Weight | 289.23 g/mol |
Appearance | White to pale yellow crystalline powder |
Solubility | Lipophilic compound, soluble in DMSO (>50 mg/ml) |
Parameter | Fexinidazole | Nifurtimox | Eflornithine |
---|---|---|---|
Administration Route | Oral | Oral | Intravenous |
Treatment Duration | 10 days | 60 days | 14 days |
CNS Penetration | High | Moderate | Low |
Stage Coverage | Both stages | Early stage | Late stage |
Parameter | Details |
---|---|
Location | Democratic Republic of Congo (2020-2022) |
Patient Cohort | 1,742 stage II HAT patients |
Treatment Outcome | 94.3% cure rate at 18-month follow-up |
Adverse Events | 8.2% reported mild gastrointestinal symptoms |
Parameter | Details |
---|---|
Organization | Doctors Without Borders (MSF) |
Implementation | Field deployment across 23 treatment centers |
Operational Impact | Reduced treatment costs by 62% vs. previous protocols |
Logistical Benefit | Eliminated cold chain requirements |
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