Complete Guide to 2-Methoxypyridine-4-boronic Acid
Table of Contents
1. Product Overview & Specifications
| Parameter | Specification |
|---|---|
| CAS Number | 1072931-77-4 |
| Molecular Formula | C₆H₈BNO₃ |
| Molecular Weight | 168.95 g/mol |
| Purity | ≥97% (HPLC) |
| Appearance | White to off-white crystalline powder |
| Storage Conditions | 2-8°C in inert atmosphere |
2. Key Applications & Industrial Uses
Pharmaceutical Development
Critical intermediate for kinase inhibitors and anticancer agents
Organic Synthesis
Suzuki-Miyaura cross-coupling reactions for aryl-aryl bond formation
Material Science
Building block for OLED materials and conductive polymers
3. Technical Comparison with Similar Compounds
| Compound | Reactivity | Solubility | Typical Yield |
|---|---|---|---|
| 2-Methoxypyridine-4-boronic acid | High | Soluble in THF, DMF | 85-92% |
| 4-Methoxyphenylboronic acid | Moderate | Soluble in EtOH | 75-82% |
| 3-Methoxypyridine-5-boronic acid | Low | Partial in DCM | 60-68% |
4. Detailed Usage Scenarios
Scenario 1: Suzuki Coupling in Drug Synthesis
Reaction conditions: Pd(PPh3)4 catalyst, Na2CO3 base, DME/H2O solvent system at 80°C
Scenario 2: Material Polymerization
Co-polymerization with thiophene derivatives for conductive materials
5. Verified Customer Case Studies
Case Study 1: PharmaSynth Co., Ltd. (2024)
Application: Developed novel kinase inhibitor using 50kg batch
Result: Achieved 89% coupling efficiency in final API synthesis
Case Study 2: MaterialInnovate Inc. (2023)
Application: OLED emitter material development
Result: 15% improvement in device efficiency vs previous formulations
6. Procurement & Inquiry Guidance
Available package sizes: 1g, 5g, 25g, 100g, 1kg
Lead time: 2-3 weeks for standard orders
Contact technical team:
- Email: info@vivalr.com
- Tel: (86) 15866781826
Request SDS and COA documents for batch-specific analysis


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